A process for the preparation of ziprasidone and a novel intermediate useful in its preparation. The process comprises the reduction of a compound (III) to give a compound (V) which is then reduced to compound (II). This is reacted with compound (IV) to give the desired compound.
申请公布号
EP1787990(A2)
申请公布日期
2007.05.23
申请号
EP20060023525
申请日期
2006.11.13
申请人
DIPHARMA FRANCIS S.R.L.;LUNDBECK PHARMACEUTICALS ITALY
发明人
ZANON, JACOPO;MARTINI, OSCAR;CIARDELLA, FRANCESCO;GREGORI, LUCA;SBROGIO, FEDERICO;CASTELLIN, ANDREA
