发明名称 AN IMPROVED PROCESS FOR THE PREPARATION OF GRANISETRON HYDROCHLORIDE
摘要 The present invention relates to an improved process for the preparation of Granisetron hydrochloride of formula (I). More particularly this invention relates to the preparation of Granisetron hydrochloride using methyl isobutyl ketone (MIBK) as a single solvent in presence of an organic base such as triethylamine.
申请公布号 WO2007054784(A1) 申请公布日期 2007.05.18
申请号 WO2006IB03146 申请日期 2006.11.08
申请人 ORCHID CHEMICALS & PHARMACEUTICALS LIMITED;SHARMA, HITESH, CHANDRAPRAKASH;RAO, SIRIPRAGADA, MAHENDER;KUMAR, SHANMUGA, SUNDARAM, BHARANI 发明人 SHARMA, HITESH, CHANDRAPRAKASH;RAO, SIRIPRAGADA, MAHENDER;KUMAR, SHANMUGA, SUNDARAM, BHARANI
分类号 C07D451/14;C07C69/14;C07D471/08 主分类号 C07D451/14
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