发明名称 |
METHOD OF MODULATING THE PROLIFERATION OF MEDULLARY THYROID CARCINOMA CELLS |
摘要 |
<p>The present invention is directed to a compound of the formula:
€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ cyclo[Tic-Tyr-D-Trp-Lys-Abu-Phe];
€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ D-Nal-cyclo[Cys-Tyr-D-Trp-Lys-Val-Cys]-Thr-NH 2 ;
€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ 4-(2-Hydroxyethyl)-1-piperazinylacetyl-D-Phe-cyclo(Cys-Tyr-D-Trp-Lys-Abu-Cys)-Thr-NH 2 ; and
€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ 4-(2-Hydroxyethyl)-1-piperazine-2-ethanesulfonyl-D-Phe-cyclo(Cys-Tyr-D-Trp-Lys-Abu-Cys)-Thr-NH 2 ,</p> |
申请公布号 |
EP1390406(B1) |
申请公布日期 |
2007.05.16 |
申请号 |
EP20020725077 |
申请日期 |
2002.03.06 |
申请人 |
IL CONSORZIO FERRARA RICHERCHE;SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES S.A.S. |
发明人 |
DEGLI UBERTI, ETTORE, CIRO;ZATELLI, MARIA, CHIARA;CULLER, MICHAEL, DEWITT |
分类号 |
C07K14/655;G01N33/48;A61K38/00;A61K38/08;A61K38/31;A61K45/00;A61K51/00;A61P35/00;A61P35/04;A61P43/00;C07K7/06;C07K7/64;C12N5/06;C12Q1/02;G01N33/68 |
主分类号 |
C07K14/655 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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