发明名称 Process for production of 1-aryl-5-(trifluoromethyl)-1h-tetrazoles
摘要 The present invention relates to a process for producing an N-aryl-2,2,2-trifluoroacetimidoyl chloride represented by Formula (2): the process comprising the step of reacting in an organic solvent a tertiary amine, a 2,2,2-trifluoro-N-arylacetamide represented by Formula (1): and at least one member selected from the group consisting of phosphorus oxychloride and diphenyl chlorophosphate; and a process for producing a 1-aryl-5-(trifluoromethyl)-1H-tetrazole represented by Formula (4): the process comprising the step of reacting in an aromatic hydrocarbon solvent, in the presence of an amine salt, an N-aryl-2,2,2-trifluoroacetimidoyl chloride represented by Formula (2) shown above and an azide.
申请公布号 US2007106080(A1) 申请公布日期 2007.05.10
申请号 US20040573034 申请日期 2004.09.30
申请人 TOYO KASEI KOGYO COMPANY LIMITED 发明人 HAGIYA KAZUTAKE;SATO YASUHIRO;KOGURO KIYOTO;MITSUI SUNAO
分类号 C07D257/04;C07C249/02;C07C257/02 主分类号 C07D257/04
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