发明名称 CHROMAN COMPOUNDS AS 5-HT1B ANTAGONISTS
摘要 <p>Chroman derivatives according to formula (I), wherein R&lt;SUP&gt;1&lt;/SUP&gt;, R&lt;SUP&gt;2&lt;/SUP&gt;, R&lt;SUP&gt;3&lt;/SUP&gt; and R&lt;SUP&gt;4&lt;/SUP&gt; are as defined in the specification, pharmaceutically-acceptable salts, methods of making, pharmaceutical compositions containing and methods for using the same. The compounds are 5-HT&lt;SUB&gt;1B&lt;/SUB&gt; antagonists and are useful in the treatment of mood and anxiety disorders .as well as cognitive disorders.</p>
申请公布号 WO2007053095(A1) 申请公布日期 2007.05.10
申请号 WO2006SE01254 申请日期 2006.11.03
申请人 ASTRAZENECA AB;BERNSTEIN, PETER;HILL, DANIEL;NUGIEL, DAVID;PIERSON, EDWARD;SHENVI, ASHOKKUMAR;JACOBS, ROBERT 发明人 BERNSTEIN, PETER;HILL, DANIEL;NUGIEL, DAVID;PIERSON, EDWARD;SHENVI, ASHOKKUMAR;JACOBS, ROBERT
分类号 C07D311/66;A61K31/353;A61P25/18;A61P25/22;A61P25/24;A61P25/28 主分类号 C07D311/66
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