发明名称 |
LINEAR BASIC COMPOUNDS HAVING NK-2 ANTAGONIST ACTIVITY AND FORMULATIONS THEREOF |
摘要 |
Described herein are compounds of formula (I) useful as antagonists of tachykinins in general, and in particular of neurokinin A; and the pharmaceutical formulations comprising the compounds of formula (I).
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申请公布号 |
RS36504(A) |
申请公布日期 |
2007.04.10 |
申请号 |
YU2004P000365 |
申请日期 |
2002.10.28 |
申请人 |
MALESCI ISTITUTO FARMACOBIOLOGICO S.P.A., VIA LUNGO L EMA 7 |
发明人 |
SISTO ALESSANDRO;CACIAGLI VALERIO;ALTAMURA MARIA;GIOLITTI ALESSANDRO;FEDI VALENTINA;GUIDI ANTONIO;GIANNOTTI DANILO;HARMAT NICHOLAS;NANNICINI ROSSANO;PASQUI FRANCO;MAGGI CARLO ALBERTO |
分类号 |
A61K38/00;C07K5/062;A61K31/38;A61K31/425;A61K38/05;A61P1/00;A61P1/04;A61P9/00;A61P11/06;A61P13/02;A61P15/10;A61P17/00;A61P17/06;A61P19/02;A61P25/00;A61P25/02;A61P25/04;A61P25/18;A61P25/22;A61P25/24;A61P27/02;A61P27/14;A61P27/16;A61P29/00;A61P31/18;A61P35/00;A61P37/00;A61P37/06;A61P37/08;A61P43/00;C07D333/38;C07D333/70;C07D409/12;C07D413/12;C07D417/12;C07K5/06;C07K5/065 |
主分类号 |
A61K38/00 |
代理机构 |
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