发明名称 Crystalline and amorphous pyrimidine compounds and processes for preparing pyrimidine compounds
摘要 Crystals of 5-[2-amino-4-(2-furyl)pyrimidin-5-yl]-1-methylpyridin-2(1H)-one having a diffraction peak at a diffraction angle (2theta±0.2°) of 9.7° and/or 21.9° in a powder X-ray diffraction are suitable for an active ingredient of a preventing and therapeutic agent for diseases such as constipation. Crystals of 5-[2-amino-4-(2-furyl)pyrimidin-5-yl]-1-methylpyridin-2(1H)-one hydrate and amorphous 5-[2-amino-4-(2-furyl)pyrimidin-5-yl]-1-methylpyridin-2(1H)-one hydrate are also suitable for an active ingredient of a preventing and therapeutic agent for diseases such as constipation.
申请公布号 US2007078151(A1) 申请公布日期 2007.04.05
申请号 US20060378307 申请日期 2006.03.20
申请人 EISAI CO., LTD. 发明人 HARADA HITOSHI;ISHIHARA HIROSHI;SATO YOSHIAKI;CHIBA HIROYUKI;KOMATSU YUKI;INOUE SUSUMU;OZEKI NAOKI
分类号 A61K31/506;C07D405/14 主分类号 A61K31/506
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