发明名称 INDOLE DERIVATIVES USEFUL A.O. FOR THE TREATMENT OF OSTEOPOROSIS
摘要 A COMPOUND OF FORMULA (1) OR A SALT THEREOF, OR A SOLVATE THEREOF, WHEREIN; R1 AND R2 EACH INDEPENDENTLY REPRESENTS C1-6ALKOXY OR HALO; R3 AND R4 EACH INDEPENDENTLY REPRESENTS HYDROGEN, C1-6ALKOXY, ARYLC1-6ALKOXY, HYDROXY, CARBOXYC1-6ALKOXY, HYDROXYC1-6ALKOXY, DIHYDROXYC1-6ALKOXY, MONO-AND DI-(C1-6ALKYL)AMINO C1-6ALKOXY OR AMINOC1-6ALKOXY, AND; R5 REPRESENTS -NRSRT WHEREIN RS AND RT EACH INDEPENDENTLY REPRESENT HYDROGEN, UNSUBSTITUTED OR SUBSTITUTED C1-6ALKYL, OR UNSUBSTITUTED OR SUBSTITUTED HETEROCYCLYL, A PROCESS FOR THE PREPARATION OF SUCH A COMPOUND, A PHARMACEUTICAL COMPOSITION CONTAINING SUCH A COMPOUND AND THE USE OF THE COMPOUND OR COMPOSITION IN MEDICINE.
申请公布号 MY129425(A) 申请公布日期 2007.03.30
申请号 MYPI20002728 申请日期 2000.06.16
申请人 NIKEM RESEARCH S.R.L 发明人 FARINA, DR CARLO;GAGLIARDI, DR STEFANIA;NOVELLA PIETRO A T
分类号 C07D401/12;A61K31/404;A61K31/4439;A61K31/454;A61K31/496;A61K31/506;A61P1/00;A61P1/04;A61P3/06;A61P9/10;A61P11/00;A61P13/12;A61P17/00;A61P17/06;A61P19/02;A61P19/10;A61P25/28;A61P27/02;A61P29/00;A61P31/04;A61P31/12;A61P31/16;A61P31/18;A61P35/00;A61P35/02;A61P37/06;A61P43/00;C07D209/18;C07D403/12 主分类号 C07D401/12
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