发明名称 |
N-ALKANOYLPHENYLALANINE DERIVATIVES |
摘要 |
COMPOUDS OF THE FORMULA :(FORMULA 1) AS WELL AS THEIR SALTS AND ESTERS ARE DISCLOSED WHEREIN X, X', Z, AND Y ARE AS DESCRIBED IN THE SPECIFICATION AND WHICH HAVE ACTIVITY AS INHIBITORS OF BINDING BETWEEN VCAM-1 AND CELLS EXPRESSING VLA-4. SUCH COMPOUNDS ARE USEFUL FOR TREATING DISEASES WHOSE SYMPTOMS AND/OR DAMAGE ARE RELATED TO THE BINDING OF VCAM-1 TO CELLS EXPRESSING VLA-4.
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申请公布号 |
MY129295(A) |
申请公布日期 |
2007.03.30 |
申请号 |
MYPI9803840 |
申请日期 |
1998.08.21 |
申请人 |
F. HOFFMANN-LA ROCHE AG |
发明人 |
LI CHEN;ROBERT WILLIAM GUTHRIE;TAI-NANG HUANG;KENNETH G. HULL;ACHYTHARAO SIDDURI;JEFFERSON WRIGHT TILLEY |
分类号 |
C07C233/87;A61K31/165;A61K31/198;A61K31/33;A61K31/357;A61K31/36;A61K31/401;A61K31/41;A61K31/415;A61K31/4166;A61K31/42;A61K31/426;A61K31/44;A61K31/4409;A61K31/4418;A61K31/4427;A61K31/4439;A61K31/47;A61K31/496;A61K31/505;A61K31/519;A61K31/5375;A61K31/5377;A61P1/00;A61P11/06;A61P19/02;C07C233/81;C07C235/40;C07C235/52;C07C235/64;C07C235/82;C07C237/24;C07C237/36;C07C255/41;C07C255/57;C07C271/22;C07C275/18;C07C275/24;C07C275/30;C07C275/60;C07C317/44;C07C317/50;C07C323/39;C07C323/60;C07C335/08;C07D207/16;C07D211/64;C07D213/81;C07D213/82;C07D213/89;C07D215/50;C07D217/26;C07D231/14;C07D233/32;C07D233/38;C07D239/28;C07D249/06;C07D257/04;C07D261/08;C07D261/18;C07D277/14;C07D277/20;C07D277/56;C07D295/08;C07D295/088;C07D295/14;C07D317/30;C07D317/68;C07D401/06;C07D487/04 |
主分类号 |
C07C233/87 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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