发明名称 |
Tricyclic quinolinone and tricyclic quinoline androgen receptor modulator compounds and methods |
摘要 |
Non-steroidal tricyclic quinolinone and tricyclic quinoline compounds and compositions that are agonists, partial agonists and/or antagonists for androgen receptors (AR), their preparation and their uses are described.
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申请公布号 |
US2007072849(A1) |
申请公布日期 |
2007.03.29 |
申请号 |
US20060601251 |
申请日期 |
2006.11.17 |
申请人 |
HIGUCHI ROBERT I;ZHI LIN;KARANEWSKY DONALD S;THOMPSON ANTHONY W;CAFERRO THOMAS R;MANI NEELAKANDHA S;CHEN JYUN-HUNG;CUMMINGS MARQUIS L;EDWARDS JAMES P;ADAMS MARK E;DECKHUT CHARLOTTE L |
发明人 |
HIGUCHI ROBERT I.;ZHI LIN;KARANEWSKY DONALD S.;THOMPSON ANTHONY W.;CAFERRO THOMAS R.;MANI NEELAKANDHA S.;CHEN JYUN-HUNG;CUMMINGS MARQUIS L.;EDWARDS JAMES P.;ADAMS MARK E.;DECKHUT CHARLOTTE L. |
分类号 |
A61K31/542;G01N33/50;A61K31/498;A61K31/5383;A61P5/00;A61P5/26;A61P5/28;A61P13/08;A61P15/08;A61P15/10;A61P17/00;A61P17/10;A61P17/14;A61P19/10;A61P35/00;A61P43/00;C07D487/02;C07D498/02;C07D498/04;C07D498/14 |
主分类号 |
A61K31/542 |
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