PROCESS FOR PREPARING BENZAZEPINE COMPOUNDS OR SALTS THEREOF

摘要

This invention provides a process for preparing benzazepine compounds of the formula (1): wherein X¹is a halogen atom, R¹and R²are a lower alkyl group, or salts thereof as well as intermediate benzoic acid compounds in high yield and high purity on industrial scale, which are useful as an intermediate for preparing a pharmaceutically active 2,3,4,5-tetrahydro-1H-1-benzazepine compound having vasopressin antagonistic activity.