发明名称 |
PYRIDAZINONE DERIVATIVES USED FOR THE TREATMENT OF PAIN |
摘要 |
A pyridazinone derivative compound shown by the following formula (I): where in R1 is selected from hydrogen, etc.; R2 is selected from substituted or unsubstituted aryl, etc.; R3 is hydrogen, etc.;p is 0, 1 or 2; R4 and R5 are each hydrogen, etc.; R6 and R7 are taken together to form a group of the formula: wherein R8 is hydrogen; X is selected from oxygen, etc; R10 is selected from hydrogen, etc.; R11 is selected from hydrogen, etc.; R12 is selected from hydrogen, etc.; R13 is selected from hydrogen, etc.; R14 is selected from hydrogen, etc.; m and n are each 0, 1, or 2, or a pharmaceutically acceptable salt thereof, which is useful as a medicament.</ SDOAB>
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申请公布号 |
CA2620740(A1) |
申请公布日期 |
2007.03.08 |
申请号 |
CA20062620740 |
申请日期 |
2006.08.31 |
申请人 |
WAKUNAGA PHARMACEUTICAL CO., LTD.;ASTELLAS PHARMA INC. |
发明人 |
YOKOMOTO, MASAHARU;MIZUHARA, HIDEKAZU;KASAHARA, CHIYOSHI;KINOSHITA, TOMOHIKO;YAMAZAKI, HITOSHI;MISUMI, KEIJI;KUBOTA, HIROKAZU;ASANO, TORU;KONTANI, TORU |
分类号 |
C07D487/04;A61K31/495;A61P29/00;C07D487/20 |
主分类号 |
C07D487/04 |
代理机构 |
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