发明名称 THIAZOLE DERIVATIVE
摘要 <p>[PROBLEMS] To provide a compound which is useful as a GK activator. [MEANS FOR SOLVING PROBLEMS] As a result of an extensive study on thiazole derivatives, it is found that a compound having an oxamoyl group, a glycol group or the like on a thiazole ring and a compound having an acetamide group substituted by a dicyclic heteroaryl group such as a quinolyl have a good GK activation effect. These compounds are useful as therapeutic agents for diabetes, particularly type 2 diabetes.</p>
申请公布号 WO2007026761(A1) 申请公布日期 2007.03.08
申请号 WO2006JP317102 申请日期 2006.08.30
申请人 ASTELLAS PHARMA INC.;HAYAKAWA, MASAHIKO;NIGAWARA, TAKAHIRO;TSUCHIYA, KAZUYUKI;ISHIBASHI, NAOKI;OKUMURA, MITSUAKI;KAWAMOTO, YUICHIRO;NAGAYOSHI, AKIRA 发明人 HAYAKAWA, MASAHIKO;NIGAWARA, TAKAHIRO;TSUCHIYA, KAZUYUKI;ISHIBASHI, NAOKI;OKUMURA, MITSUAKI;KAWAMOTO, YUICHIRO;NAGAYOSHI, AKIRA
分类号 C07D277/20;A61K31/426;A61K31/4709;A61K31/517;A61P3/10;A61P43/00;C07D277/44;C07D277/56;C07D417/04;C07D417/12 主分类号 C07D277/20
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