发明名称 2,3,4,5-TETRAHYDRO-1H-BENZO[d]AZEPINES SUBSTITUEES EN POSITION 6 COMME AGONISTES DES RECEPTEURS 5-HT2C
摘要 The present invention provides 6-substituted 2,3,4,5-tetrahydro-1H-benzo[d]azepines of Formula I as selective 5-HT 2C receptor agonists for the treatment of 5-HT 2C associated disorders including obesity, obsessive/compulsive disorder, depression, and anxiety: where: R 6 is -S-L-R 15 and other substituents are as defined in the specification.
申请公布号 MA28486(B1) 申请公布日期 2007.03.01
申请号 MA20060029343 申请日期 2006.09.25
申请人 ELI LILLY AND COMPANY 发明人 ALLEN, JOHN, GORDON;BRINER, KARIN;COHEN, MICHAEL, PHILIP;GALKA, CHRISTOPHER, STANLEY;HELLMAN, SARAH, LYNNE;MARTINEZ-GRAU, MARIA, ANGELES;REINHARD, MATTHEW, ROBERT;RODRIGUEZ, MICHAEL, JOHN;ROTHHAAR, ROGER, RYAN;TIDWELL, MICHAEL, WADE;VICTOR, FRANTZ;WILLIAMS, ANDREW, CAERWYN;ZHANG, DEYI;BOYD, STEVEN, ARMEN;CONWAY, RICHARD, GERARD;DEO, ARUNDHATI, S.;LEE, WAI-MAN;SIEDEM, CHRISTOPHER, STEPHEN;SINGH, AJAY;MAZANETZ, MICHAEL, PHILIP;ELI LILLY AND COMPANY
分类号 C07D223/16;C07D401/12;C07D403/06;C07D403/12;C07D405/12;C07D409/12;C07D413/12;C07D413/14;C07D417/06;C07D417/12;(IPC1-7):C07D223/16 主分类号 C07D223/16
代理机构 代理人
主权项
地址