发明名称 Fused benzene derivative and use
摘要 Disclosed are compounds of formula (I) wherein the substituents are as described in the specification. Fused benzene derivatives as disclosed are androgen receptor agonists and are useful for the treatment of hypogonadism, climacteric disturbance, osteoporosis and hormone-resistant cancer.
申请公布号 NZ538713(A) 申请公布日期 2007.01.26
申请号 NZ20030538713 申请日期 2003.08.11
申请人 TAKEDA CHEMICAL INDUSTRIES, LTD 发明人 SHIRAISHI, MITSURU;HARA, TAKAHITO;KANZAKI, NAOYUKI;YAMAMOTO, SATOSHI;MIYAWAKI, TOSHIO;KUSAKA, MASAMI
分类号 A61P5/26;A61P13/08;A61P15/00;A61P15/10;A61P15/12;A61P19/10;A61P35/00;A61P43/00;C07C35/52;C07C217/04;C07C255/52;C07C255/53;C07C255/54;C07C255/56;C07D207/06;C07D207/08;C07D207/10;C07D207/12;C07D207/14;C07D207/16;C07D207/22;C07D207/24;C07D209/46;C07D211/22;C07D211/28;C07D211/34;C07D211/42;C07D211/46;C07D211/60;C07D211/62;C07D211/74;C07D231/08;C07D261/04;C07D265/02;C07D267/10;C07D295/073;C07D295/112;C07D295/155;C07D303/46;C07D307/79;C07D333/54;C07D405/04;C07D409/04;C07D491/10;C07D491/113;(IPC1-7):C07C35/52;C07D209/44;C07D211/14;C07D217/04;C07D231/04;C07D231/06;C07D295/06;C07D295/14;C07D307/81;A61K31/045;A61K31/277;A61K31/336;A61K31/402;A61K31/403;A61K31/42;A61K31/438;A61K31/445;A61K31/451;A61K31/452;A61K31/453;A61K31/472;A61K31/495;A61K31/535;A61K31/537;A61K31/54;A61K31/55;A61K31/553;A61K31/45 主分类号 A61P5/26
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