发明名称 |
Fused benzene derivative and use |
摘要 |
Disclosed are compounds of formula (I) wherein the substituents are as described in the specification. Fused benzene derivatives as disclosed are androgen receptor agonists and are useful for the treatment of hypogonadism, climacteric disturbance, osteoporosis and hormone-resistant cancer.
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申请公布号 |
NZ538713(A) |
申请公布日期 |
2007.01.26 |
申请号 |
NZ20030538713 |
申请日期 |
2003.08.11 |
申请人 |
TAKEDA CHEMICAL INDUSTRIES, LTD |
发明人 |
SHIRAISHI, MITSURU;HARA, TAKAHITO;KANZAKI, NAOYUKI;YAMAMOTO, SATOSHI;MIYAWAKI, TOSHIO;KUSAKA, MASAMI |
分类号 |
A61P5/26;A61P13/08;A61P15/00;A61P15/10;A61P15/12;A61P19/10;A61P35/00;A61P43/00;C07C35/52;C07C217/04;C07C255/52;C07C255/53;C07C255/54;C07C255/56;C07D207/06;C07D207/08;C07D207/10;C07D207/12;C07D207/14;C07D207/16;C07D207/22;C07D207/24;C07D209/46;C07D211/22;C07D211/28;C07D211/34;C07D211/42;C07D211/46;C07D211/60;C07D211/62;C07D211/74;C07D231/08;C07D261/04;C07D265/02;C07D267/10;C07D295/073;C07D295/112;C07D295/155;C07D303/46;C07D307/79;C07D333/54;C07D405/04;C07D409/04;C07D491/10;C07D491/113;(IPC1-7):C07C35/52;C07D209/44;C07D211/14;C07D217/04;C07D231/04;C07D231/06;C07D295/06;C07D295/14;C07D307/81;A61K31/045;A61K31/277;A61K31/336;A61K31/402;A61K31/403;A61K31/42;A61K31/438;A61K31/445;A61K31/451;A61K31/452;A61K31/453;A61K31/472;A61K31/495;A61K31/535;A61K31/537;A61K31/54;A61K31/55;A61K31/553;A61K31/45 |
主分类号 |
A61P5/26 |
代理机构 |
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代理人 |
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