摘要 |
The invention relates to compound of the formula (I) or its salt, wherein -R<SUP>1</SUP>, -R<SUP>2</SUP>, -R<SUP>3</SUP>, -R<SUP>4</SUP>, -R<SUP>5</SUP>, -M-, -X- and -Y= are as defined in the description, their use of as, medicament, the process for their preparation and use for the treatment of JAK3 mediated diseases. |
申请人 |
ASTELLAS PHARMA INC.;INOUE, TAKAYUKI;TOJO, TAKASHI;MORITA, MASATAKA;NAKAJIMA, YUTAKA;HATANAKA, KEIKO;SHIRAKAMI, SHOHEI;SASAKI, HIROSHI;TANAKA, AKIRA;TAKAHASHI, FUMIE;MUKOYOSHI, KOICHIRO;HIGASHI, YASUYUKI;OKIMOTO, AKIRA;HONDO, TAKESHI;SAWADA, HITOSHI |
发明人 |
INOUE, TAKAYUKI;TOJO, TAKASHI;MORITA, MASATAKA;NAKAJIMA, YUTAKA;HATANAKA, KEIKO;SHIRAKAMI, SHOHEI;SASAKI, HIROSHI;TANAKA, AKIRA;TAKAHASHI, FUMIE;MUKOYOSHI, KOICHIRO;HIGASHI, YASUYUKI;OKIMOTO, AKIRA;HONDO, TAKESHI;SAWADA, HITOSHI |