发明名称 2-AMINO-QUINAZ0LIN-5-ONES AS HSP90 INHIBITORS USEFUL IN TREATING PROLIFERATION DISEASES
摘要 2-Amino-quinazolin-5-one compounds, stereoisomers, tautomers, pharmaceutically acceptable salts, and prodrugs thereof; compositions that include a pharmaceutically acceptable carrier and one or more of the 2-amino-quinazolin-5-one compounds, either alone or in combination with at least one additional therapeutic agent. Methods of using the 2-amino-quinazolin-5-one compounds, either alone or in combination with at least one additional therapeutic agent, in the prophylaxis or treatment of cell proliferative diseases.
申请公布号 WO2006113498(A3) 申请公布日期 2007.01.11
申请号 WO2006US14194 申请日期 2006.04.14
申请人 CHIRON CORPORATION;MACHAJEWSKI, TIMOTHY, D.;GAO, ZHENHAI;LEVINE, BARRY, H.;ANTONIOS-MCCREA, WILLIAM;BELLAMACINA, CORNELIA, R.;COSTALES, ABRAN;DOUGHAN, BRANDON, M.;FONG, SUSAN;HENDRICKSON, THOMAS;LIN, XIAODONG;MCBRIDE, CHRISTOPHER;MCKENNA, MAUREEN;RICO, ALICE, C.;SHAFER, CYNTHIA, M.;WANG, X., MICHAEL;ZHOU, YASHEEN;XIA, YI;MENDENHALL, KRIS, G. 发明人 MACHAJEWSKI, TIMOTHY, D.;GAO, ZHENHAI;LEVINE, BARRY, H.;ANTONIOS-MCCREA, WILLIAM;BELLAMACINA, CORNELIA, R.;COSTALES, ABRAN;DOUGHAN, BRANDON, M.;FONG, SUSAN;HENDRICKSON, THOMAS;LIN, XIAODONG;MCBRIDE, CHRISTOPHER;MCKENNA, MAUREEN;RICO, ALICE, C.;SHAFER, CYNTHIA, M.;WANG, X., MICHAEL;ZHOU, YASHEEN;XIA, YI;MENDENHALL, KRIS, G.
分类号 C07D239/84;A61K31/517;A61P35/00;C07D401/04;C07D401/10;C07D403/04;C07D403/10;C07D403/12;C07D413/10;C07D417/10;C07D417/12 主分类号 C07D239/84
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