发明名称 PROCESS FOR THE PREPARATION OF 5-(1-PIPERAZINYL) BENZOFURAN-2-CARBOXAMIDE BY TRANSITION METAL-CATALYSED AMINATION
摘要 <p>PROCESS FOR THE PREPARATION OF 5-(1-PIPERAZINYL)BENZOFURAN-2-CARBOXAMIDE IN WHICH , AS INTERMEDIATE STEP, 5-BROMOSALICYLALDEHYDE OR ONE OF ITS DERIVATIVES IS REACTED IN A TRANSITION METAL-CATALYSED AMINATION WITH R²-PIPERAZINE, IN WHICH R² IS AS DEFINED IN CLAIM 1.</p>
申请公布号 MY127851(A) 申请公布日期 2006.12.29
申请号 MY2000PI05614 申请日期 2000.11.30
申请人 MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG 发明人 BATHE, ANDREAS;EMMERT, STEFFEN;HELFERT, BERND;BOTTCHER, HENNING
分类号 C07D295/08;C07D295/112;C07B61/00;C07D295/04;C07D295/10;C07D295/20;C07D295/205;C07D295/28;C07D307/85;C07D405/00;C07D405/04 主分类号 C07D295/08
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