发明名称 TRIAZOLOPYRIDINE DERIVATIVES AS CANNABINOID RECEPTOR 1 ANTAGONISTS
摘要 <p>The present application describes compounds according to Formula I, pharmaceutical compositions comprising at least one compound according to Formula I and optionally one or more additional therapeutic agents, and methods of treatment using the compounds according to Formula I both alone and in combination with one or more additional therapeutic agents. The compounds have the following general formula I including all solvates, pharmaceutically acceptable salts and stereoisomers, wherein R&lt;SUP&gt;1&lt;/SUP&gt; , R&lt;SUP&gt;2&lt;/SUP&gt;, R&lt;SUP&gt;3&lt;/SUP&gt;, R&lt;SUP&gt;4&lt;/SUP&gt; and R&lt;SUP&gt;5&lt;/SUP&gt; are described herein. '</p>
申请公布号 WO2006138695(A1) 申请公布日期 2006.12.28
申请号 WO2006US23716 申请日期 2006.06.19
申请人 BRISTOL-MYERS SQUIBB COMPANY;SUN, CHONGQING;SHER, PHILIP M.;WU, GANG;EWING, WILLIAM R.;HUANG, YANTING;LEE, TAEKYU;MURUGESAN, NATESAN;SULSKY, RICHARD B. 发明人 SUN, CHONGQING;SHER, PHILIP M.;WU, GANG;EWING, WILLIAM R.;HUANG, YANTING;LEE, TAEKYU;MURUGESAN, NATESAN;SULSKY, RICHARD B.
分类号 C07D471/04;A61K31/435;A61P25/00;A61P37/00 主分类号 C07D471/04
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