发明名称 CARBOXAMIDE INHIBITORS OF TGFB
摘要 Pyrimidine having a pyridylamine group at C- 4 of the pyrimidine and an amide group on the pyridine ring (compounds of formula I) are useful in the treatment of conditions associated with excessive TGFB activity.
申请公布号 WO2006105222(A3) 申请公布日期 2006.12.28
申请号 WO2006US11509 申请日期 2006.03.27
申请人 SCIOS INC.;AXON, JONATHAN;CHAKRAVARTY, SARVAJIT;HART, BARRY;MCENROE, GLENN;MURPHY, ALISON;PONTIUS, KAREN;SHENG, PEIJUE;WANG, XIAOJING;YELLAPREGADA, SHANTHI 发明人 AXON, JONATHAN;CHAKRAVARTY, SARVAJIT;HART, BARRY;MCENROE, GLENN;MURPHY, ALISON;PONTIUS, KAREN;SHENG, PEIJUE;WANG, XIAOJING;YELLAPREGADA, SHANTHI
分类号 C07D401/12;A61K31/506;A61K31/5377;A61P11/00;A61P35/00;C07D401/14;C07D407/14;C07H7/06;C07H13/04;C07H15/04;C07H15/18;C07H15/26 主分类号 C07D401/12
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