发明名称 Macrocyclic compounds useful as pharmaceuticals
摘要 The present invention provides compounds having formula (I), and additionally provides methods for the synthesis thereof and methods for the use thereof in the treatment of various disorders including inflammatory or autoimmune disorders, and disorders involving malignancy or increased angiogenesis, wherein R 1 -R 11 , t, X, Y, Z and n are as defined herein.
申请公布号 ZA200407156(B) 申请公布日期 2006.12.27
申请号 ZA20040007156 申请日期 2004.09.07
申请人 EISAI CO. LTD. 发明人 BOIVIN, ROCH;DU, HONG;GOTO, MASAKI;JIANG, YIMIN;KAWAKAMI, YOSHIYUKI;KUBOI, YOSHIKAZU;MATSUSHIMA, TOMOHIRO;SHEN, YONG-CHUN;WANG, YONG-CHUN;WANG, JOHN (YUAN);GUSOVSKY, FABIAN;CHIBA, KENICHI;EGUCHI, YOSHIHITO;HARMANGE, JEAN-CHRISTOPHE;KAWADA, MEGUMI;KIMURA, AKIFUMI;LEMELIN, CHARLES-ANDRU;MIZUI, YOSHIHARU;SPYVEE, MARK;YAMAMOTO, SATOSHI;MURAMOTO, KENZO;CHOW, JESSE;FUJITA, MASANORI;INOUE, ATSUSHI;KAWAI, TAKATOSHI;KOTAKE, MAKOTO;LI, XIANG-YI;SAKURAI, HIDEKI;TANAKA, ISAO;YONEDA, NAOKI;SHIROTA, HIROSHI
分类号 C07D491/044;A61K;A61K31/335;A61K31/36;A61K31/365;A61K31/395;A61K31/4178;A61K31/4188;A61K31/5377;A61P;A61P1/00;A61P1/04;A61P1/16;A61P3/10;A61P7/04;A61P9/00;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P17/00;A61P17/04;A61P17/06;A61P17/16;A61P19/02;A61P19/04;A61P19/10;A61P21/04;A61P25/00;A61P25/02;A61P25/08;A61P25/28;A61P27/02;A61P29/00;A61P31/04;A61P31/18;A61P33/06;A61P35/00;A61P37/02;A61P37/06;A61P37/08;A61P43/00;C07D;C07D267/00;C07D313/00;C07D401/12;C07D405/12;C07D491/04;C07D493/04;C07D521/00 主分类号 C07D491/044
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