发明名称 |
BICYCLOESTER DERIVATIVE |
摘要 |
<p>[PROBLEMS] To provide a novel bicycloester derivative having excellent DPP-IV inhibiting activity or a pharmacologically acceptable salt thereof. [MEANS FOR SOLVING PROBLEMS] There is provided a novel bicycloester derivative of the general formula: (1) or a pharmacologically acceptable salt thereof (for example, (2S,4S)- 1-[[N-(4-ethoxycarbonylbicyclo[2.2.2]oct-1-yl)amino]acetyl]-4- fluoropyrrolidine-2-carbonitrile).</p> |
申请公布号 |
KR20060130641(A) |
申请公布日期 |
2006.12.19 |
申请号 |
KR20067015699 |
申请日期 |
2005.02.01 |
申请人 |
KYORIN PHARMACEUTICAL CO., LTD. |
发明人 |
FUKUDA YASUMICHI;ASAHINA YOSHIKAZU;OHATA KOHEI;YOKOTA KAZUYA;MURAKAMI KOJI;MATSUI TOSHIYUKI |
分类号 |
C07D207/16;A61K31/40;A61K31/4025;A61P3/10;A61P43/00;C07D405/12;C07D407/12 |
主分类号 |
C07D207/16 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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