发明名称 SUBSTITUTED N-BENZO [D] ISOXAZOL-3-YL-AMINE DERIVATIVES AS INHIBITORS OF MGLUR5, SEROTONINE (5-HT) AND NORADRENALINE RECEPTORS, AND THE USE THEREOF FOR PRODUCING MEDICAMENTS
摘要 The invention relates to substituted N-benzo[d]isoxazol-3-yl-amine derivatives of formula (I) wherein R1,R2,R3,R4 and R5 are defined as in patent claim 1. The invention also relates to the use of said compounds for producing medicaments.
申请公布号 CA2610373(A1) 申请公布日期 2006.12.14
申请号 CA20062610373 申请日期 2006.06.06
申请人 GRUENENTHAL GMBH 发明人 MERLA, BEATRIX;JAGUSCH, UTZ-PETER;SUNDERMANN, CORINNA;GERLACH, MATTHIAS;HENNIES, HAGEN-HEINRICH;HAURAND, MICHAEL;OBERBOERSCH, STEFAN;JOSTOCK, RUTH;REICH, MELANIE
分类号 C07D261/20;A61K31/423;A61P29/00;C07D413/12 主分类号 C07D261/20
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