发明名称 HISTAMINE H3-RECEPT0R LIGANDS AND THEIR THERAPEUTIC APPLICATION
摘要 <p>The present patent application concerns new compounds of formula (I) with R&lt;SUP&gt;1&lt;/SUP&gt; and R&lt;SUP&gt;2&lt;/SUP&gt; taken together with the nitrogen atom to which they are attached, form a saturated nitrogen-containing ring, A is a saturated C1 -4 alkylene and B a C3-4 alkylene or alkenylene chain; their preparation and their use as a H3 receptor ligand for treating e.g. CNS disorders like Alzheimer's disease.</p>
申请公布号 WO2006117611(A1) 申请公布日期 2006.11.09
申请号 WO2006IB01018 申请日期 2006.04.26
申请人 BIOPROJET;BERTRAND, ISABELLE;CAPET, MARC;LECOMTE, JEANNE-MARIE;LEVOIN, NICOLAS;LIGNEAU, XAVIER;POUPARDIN-OLIVIER, OLIVIA;ROBERT, PHILIPPE;SCHWARTZ, JEAN-CHARLES 发明人 BERTRAND, ISABELLE;CAPET, MARC;LECOMTE, JEANNE-MARIE;LEVOIN, NICOLAS;LIGNEAU, XAVIER;POUPARDIN-OLIVIER, OLIVIA;ROBERT, PHILIPPE;SCHWARTZ, JEAN-CHARLES
分类号 C07D295/088;A61K31/40;A61K31/445;A61P25/00;C07D307/79;C07D317/54;C07D319/18 主分类号 C07D295/088
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