发明名称 PYRAZOLOQUINOLONE DERIVATIVE AND USE THEREOF
摘要 <p>The present invention provides a pyarzoloquinolone derivative having kinase inhibitory activity. The derivative is represented by the formula: wherein R 1 is an aryl group which may be substituted, or an aromatic heterocyclic group which may be substituted; R 2 is a hydrogen atom, an amino group which may be substituted, a hydroxy group which may be substituted, or a thiol group which may be substituted; R 3 , R 4 , R 5 and R 6 , which may be identical or different, are each (1) a hydrogen atom, (2) a nitro group, (3) a cyano group, (4) a halogen atom, (5) a hydrocarbon group which may be substituted, (6) an amino group which may be substituted, (7) a hydroxy group which may be substituted, or (8) a thiol group which may be substituted; and R 3 and R 4 , R 4 and R 5 , and R 5 and R 6 may respectively form a ring together with the adjacent carbon atom, or salt thereof.</p>
申请公布号 EP1719771(A1) 申请公布日期 2006.11.08
申请号 EP20050710686 申请日期 2005.02.18
申请人 TAKEDA PHARMACEUTICAL COMPANY LIMITED 发明人 FUKUMOTO, SHOJI;YAMAMOTO, TAKESHI;OKANIWA, MASANORI;TANAKA, TOSHIMASA
分类号 C07D471/04;A61K31/4745;A61K31/496;A61K31/5377;A61P19/10;A61P35/00;A61P43/00 主分类号 C07D471/04
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