发明名称 |
New hexyloxycarbonylamino-imino-methyl-phenylamino-methyl-benzimidazole-pyridine-propionic acid-ethyl ester salts such as hydrochloride useful for the prophylaxis of vein thrombosis and stroke |
摘要 |
<p>3-[(2-{[4-(hexyloxycarbonylamino-imino-methyl)-phenylamino]-methyl}-1-methyl-1H-benzimidazole-5-carbonyl)-pyridine-2-yl-amino]propionic acid ethyl ester salts (I), selected from hydrochloride, maleate, tartrate (and its enantiomers and mixtures), salicylate, citrate and malonate, and their hydrates, are new. An independent claim is included for a pharmaceutical composition comprising (I), optionally one or more inert carriers and/or diluents. ACTIVITY : Anticoagulant; Cerebroprotective; Vasotropic. MECHANISM OF ACTION : None given.</p> |
申请公布号 |
DE102005020002(A1) |
申请公布日期 |
2006.11.02 |
申请号 |
DE20051020002 |
申请日期 |
2005.04.27 |
申请人 |
BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG |
发明人 |
SIEGER, PETER;HAUEL, NORBERT;SCHMID, ROLF |
分类号 |
C07D401/12;A61K31/4439;A61P7/02 |
主分类号 |
C07D401/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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