发明名称 |
Boronic acid salts useful in parenteral formulations for selective thrombin inhibition |
摘要 |
<p>Parenteral pharmaceutical formulations comprising base addition salts of a peptide boronic acid drug, for example of Cbz-(R)-Phe-(S)-Pro-(R)-Mpg-B(OH)2. The counter-ion to the boronate may be an alkali metal or alkaline earth metal.</p> |
申请公布号 |
SI1400245(T1) |
申请公布日期 |
2006.10.31 |
申请号 |
SI20030030345T |
申请日期 |
2003.09.09 |
申请人 |
TRIGEN LIMITED |
发明人 |
MADGE DAVID JONATHAN;DOLMAN MARK;COMBE-MARZELLE SOPHIE-MARIE;KENNEDY ANTHONY JAMES;KAKKAR SANJAY KUMAR;DEADMAN JOHN JOSEPH;WALTER ARMIN;OLBRICH ALFRED;KRIMMER DIETER;WEILAND-WEIBEL ANDREA MARIA THERESIA |
分类号 |
A61K31/69;A61K38/00;A61K45/06;C07F5/02;C07K5/06;C07K5/065 |
主分类号 |
A61K31/69 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|