发明名称 Piperazinylcarbonylquinolines and-isoquinolines
摘要 Compound of the formula (I) in which R<SUP>1</SUP>, R<SUP>2 </SUP>and alk are as defined in Claim 1, are potent 5-HT<SUB>2A </SUB>antagonist and are suitable for the treatment of psychoses, schizophrenia, depression, neurological disorders, memory disorders, Parkinson's disease, amyotrophic lateral sclerosis, Alzheimer's disease, Hutington's disease, eating disorders, such as bulimia, anorexia nervosa, premenstrual syndrome and/or for positively influencing obsessive-compulsive disorder (OCD).
申请公布号 HK1061849(A1) 申请公布日期 2006.10.27
申请号 HK20040104840 申请日期 2004.07.06
申请人 MERCK PATENT GHBH 发明人 HENNING BOTTCHER;GERD BARTOSZYK;JURGEN HARTING;CHRISTOPH VAN AMSTERDAM;CHRISTOPH SEYFRIED
分类号 C07D;C07D403/06;A61K;A61K31/495;A61K31/496;A61K45/00;A61P;A61P21/00;A61P25/00;A61P25/14;A61P25/16;A61P25/18;A61P25/24;A61P25/28;A61P25/30;A61P29/00;A61P43/00;C07D215/48;C07D217/26 主分类号 C07D
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