发明名称 |
A PROCESS FOR THE PURIFICATION OF 10-DEACETYLBACCATINE III FROM 10-DE ACET YL-2- DEBENZOYL-2-PENTENOYLBACCATINE III |
摘要 |
<p>A process for the preparation of 10-deacetyl-7,10-bis- trichloroacetylbaccatine III with HPLC purity higher than 99% and free from 2-debenzoyl-2-pentenoylbaccatine III by purification of 10-deacetyl-7,10-bis- trichloroacetylbaccatineIII followed by alkaline hydrolysis of the protecting groups in position 7 and 10.</p> |
申请公布号 |
WO2006108561(A1) |
申请公布日期 |
2006.10.19 |
申请号 |
WO2006EP03162 |
申请日期 |
2006.04.07 |
申请人 |
INDENA S.P.A;GABETTA, BRUNO;GAMBINI, ANDREA |
发明人 |
GABETTA, BRUNO;GAMBINI, ANDREA |
分类号 |
C07D305/14;A61K31/337 |
主分类号 |
C07D305/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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