发明名称 |
Phenylsulfonyl-1,3-dihydro-2h-indole-2-one derivatives, their preparation and their therapeutic use |
摘要 |
The invention relates to compounds of formula: and also to the salts thereof with mineral or organic acids, and the solvates and/or hydrates thereof, with affinity for and selectivity towards the arginine-vasopressin V<SUB>1b </SUB>receptors and/or for the ocytocin receptors and, furthermore, for certain compounds, affinity for the V<SUB>1a </SUB>receptors. The invention also relates to the process for preparing them, to the intermediate compounds of formula (IV) that are useful for preparing them, to pharmaceutical compositions containing them and to their use for preparing medicinal products.
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申请公布号 |
US7119086(B2) |
申请公布日期 |
2006.10.10 |
申请号 |
US20040484370 |
申请日期 |
2004.01.16 |
申请人 |
SANOFI-AVENTIS |
发明人 |
DI MALTA ALAIN;GARCIA GEORGES;ROUX RICHARD;SCHOENTJES BRUNO;SERRADEIL-LE GAL CLAUDINE;TONNERRE BERNARD;WAGNON JEAN |
分类号 |
A61K31/496;A61K;A61K31/497;A61K31/501;A61K31/503;A61K31/506;A61K31/55;A61K31/551;A61P;A61P1/04;A61P1/08;A61P1/12;A61P1/14;A61P1/16;A61P3/04;A61P3/06;A61P3/08;A61P3/10;A61P3/12;A61P5/24;A61P5/38;A61P7/04;A61P9/00;A61P9/04;A61P9/08;A61P9/10;A61P9/12;A61P11/00;A61P11/06;A61P13/00;A61P13/02;A61P13/08;A61P13/12;A61P15/00;A61P15/04;A61P15/10;A61P17/02;A61P17/06;A61P19/02;A61P21/00;A61P21/02;A61P25/04;A61P25/06;A61P25/14;A61P25/16;A61P25/18;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P25/30;A61P25/34;A61P27/06;A61P27/12;A61P29/00;A61P29/02;A61P31/00;A61P35/00;A61P37/04;A61P37/08;A61P43/00;C07D;C07D401/12;C07D401/14;C07D403/12;C07D417/12;C07D417/14 |
主分类号 |
A61K31/496 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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