发明名称 Diaryl ethers as opioid receptor antagonist
摘要 A compound of the formula (I) wherein the variables X<SUB>1 </SUB>to X<SUB>10</SUB>, R<SUP>1 </SUP>to R<SUP>7 </SUP>including R<SUP>3'</SUP>, E, v, y, z, A and B are as described, or a pharmaceutically acceptable salt, solvate, enantiomer, racemate, diastereomer or mixtures thereof, useful for the treatment, prevention or amelioration of obesity and Related Diseases is disclosed.
申请公布号 US2006217372(A1) 申请公布日期 2006.09.28
申请号 US20050526960 申请日期 2005.03.03
申请人 BLANCO-PILLADO MARIA-JESUS;CHAPPELL MARK D;DE LA TORRE MARTA G;DIAZ BUEZO NURIA;FRITZ JAMES E;HOLLOWAY WILLIAM G;MATT JAMES E;MITCH CHARLES E;PEDREGAL-TERCERO CONCEPCION;WUIMBY STEVEN J;SIEGEL MILES G;SMITH DANA R;STUCKY RUSSELL D;TAKEUCHI KUMIKO;THOMAS ELIZABETH M;WOLFE CHAD N 发明人 BLANCO-PILLADO MARIA-JESUS;CHAPPELL MARK D.;DE LA TORRE MARTA G.;DIAZ BUEZO NURIA;FRITZ JAMES E.;HOLLOWAY WILLIAM G.;MATT JAMES E.;MITCH CHARLES E.;PEDREGAL-TERCERO CONCEPCION;WUIMBY STEVEN J.;SIEGEL MILES G.;SMITH DANA R.;STUCKY RUSSELL D.;TAKEUCHI KUMIKO;THOMAS ELIZABETH M.;WOLFE CHAD N.
分类号 A61K31/541;A61K31/496;A61K31/497;A61K31/501;A61K31/506;A61K31/5377;A61P3/04;C07C235/46;C07D213/38;C07D213/64;C07D213/643;C07D213/78;C07D213/81;C07D213/82;C07D217/04;C07D237/24;C07D241/24;C07D307/14;C07D333/20;C07D401/06;C07D401/12;C07D401/14;C07D403/02;C07D405/12;C07D409/12;C07D409/14;C07D413/02;C07D413/12;C07D417/02;C07D417/12;C07D417/14 主分类号 A61K31/541
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