发明名称 Synthesis of estetrol via estrone derived steroids
摘要 A process is provided for the making of estetrol starting from a 3-A-oxy-estra 1,3,5(10),15-tetraen-17-one, wherein A is a C<SUB>1</SUB>-C<SUB>5 </SUB>alkyl group, preferably a methyl group, or a C<SUB>7</SUB>-C<SUB>12 </SUB>benzylic group, preferably a benzyl group. This process is particularly suitable to industry.
申请公布号 US2006211669(A1) 申请公布日期 2006.09.21
申请号 US20050534079 申请日期 2005.11.14
申请人 VERHAAR MARK T;KOCH THOMAS;WARMERDAM ERWIN G J 发明人 VERHAAR MARK T.;KOCH THOMAS;WARMERDAM ERWIN G.J.
分类号 C07J1/00;A61K31/56 主分类号 C07J1/00
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