发明名称 ACYLATED PIPERIDIHES AS GLYCINE TRANSPORTER INHIBITORS
摘要 <p>The invention provides a compound of formula (I) or a salt or solvate thereof: wherein R&lt;SUP&gt;1&lt;/SUP&gt;, n, X, Y and Z are as defined in the specification, and uses of such compounds. The compounds inhibit GlyT1 transporters and are useful in the treatment of certain neurological and neuropsychiatric disorders, including schizophrenia.</p>
申请公布号 WO2006094842(A1) 申请公布日期 2006.09.14
申请号 WO2006EP02484 申请日期 2006.03.09
申请人 GLAXO GROUP LIMITED;BRADLEY, DANIEL, MARCUS;BRANCH, CLIVE, LESLIE;CHAN, WAI, NGOR;COULTON, STEVEN;DEAN, ANTHONY, WILLIAM;DOYLE, PAUL, MARTIN;EVANS, BRIAN;GILPIN, MARTIN, LEONARD;GOUGH, SHARON, LISA;MACRITCHIE, JACQUELINE, ANNE;MARSHALL, HOWARD, ROBERT;NASH, DAVID, JOHN;PORTER, RODERICK, ALAN;WARD, SIMON, EDWARD 发明人 BRADLEY, DANIEL, MARCUS;BRANCH, CLIVE, LESLIE;CHAN, WAI, NGOR;COULTON, STEVEN;DEAN, ANTHONY, WILLIAM;DOYLE, PAUL, MARTIN;EVANS, BRIAN;GILPIN, MARTIN, LEONARD;GOUGH, SHARON, LISA;MACRITCHIE, JACQUELINE, ANNE;MARSHALL, HOWARD, ROBERT;NASH, DAVID, JOHN;PORTER, RODERICK, ALAN;WARD, SIMON, EDWARD
分类号 C07D295/18;A61K31/445;A61K31/4523;A61K31/4525;A61K31/4545;A61P25/00;C07D209/08;C07D213/56;C07D213/74;C07D231/12;C07D295/192;C07D307/38;C07D307/54;C07D307/64;C07D333/24;C07D405/12;C07D471/04 主分类号 C07D295/18
代理机构 代理人
主权项
地址