发明名称 PREPARATION OF ACID ADDITION SALTS OF ZIPRASIDONE AND INTERMEDIATES THEREOF BY SOLID PHASE-GAS PHASE REACTIONS
摘要 A process for the preparation of an acid addition salt of ziprasidone base a nd intermediates thereof comprising exposing the ziprasidone base in solid form to a gaseous acid in a substantially dry environment.
申请公布号 CA2500667(A1) 申请公布日期 2006.09.11
申请号 CA20052500667 申请日期 2005.03.11
申请人 APOTEX PHARMACHEM INC. 发明人 MURTHY, K.S. KESHAVA;REY, ALLAN W.;HORNE, STEPHEN E.;DERDOUR, LOTFI;DATTA, PROBAL KANTI;EHLERT, MARTIN
分类号 C07D417/14 主分类号 C07D417/14
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