发明名称 Process for making risperidone and intermediates therefor
摘要 The formation of risperidone is enhanced by the use of enriched Z-isomer oxime intermediate(s) of formula (3) or (7). The oxime(s) can be isomerically enriched by a variety of techniques including the use of the novel acetic acid salt thereof, which affords, inter alia, resolution of the isomers and/or by heat conversion.
申请公布号 ZA200503698(B) 申请公布日期 2006.08.30
申请号 ZA20050003698 申请日期 2005.05.09
申请人 SYNTHON B.V. 发明人 PAVEL SLANINA;JIRI BARTL
分类号 C07D;C07D211/58;C07D471/04 主分类号 C07D
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