发明名称 3-aminoquinazolin-2,4-dione antibacterial agents
摘要 Antibacterial 3-aminoquinazolin-2,4-diones have formula (I) wherein: R<SUB>1 </SUB>and R<SUB>3 </SUB>include alkyl, alkenyl, cycloalkyl, aryl, hetero-cyclic, and heteroaryl; R<SUB>5</SUB>, R<SUB>6</SUB>, and R<SUB>8 </SUB>include H, alkyl, alkoxy, halo, NO<SUB>2</SUB>, CN, NH<SUB>2</SUB>, alkyl and dialkylamino; R<SUB>7 </SUB>includes hydrogen, alkyl, cycloalkyl, hetero-cyclic, fused heterocyclic, aryl and fused aryl; J and K are C or N; and pharmaceutically acceptable salts thereof.
申请公布号 US7094780(B1) 申请公布日期 2006.08.22
申请号 US20020182221 申请日期 2002.12.09
申请人 WARNER LAMBERT COMPANY LLC 发明人 BIRD PAUL;ELLSWORTH EDMUND LEE;NGUYEN DAI QUOC;SANCHEZ JOSEPH PETER;SHOWALTER HOWARD DANIEL HOLLIS;SINGH RAJESHWAR;STIER MICHAEL ANDREW;TRAN TUAN PHONG;WATSON BRIAN MORGAN;YIP JUDY
分类号 C07D239/92;C07D239/96;A61K31/505;A61K31/517;A61K31/519;A61K31/5383;A61P31/04;A61P31/14;C07D401/04;C07D403/04;C07D403/14;C07D409/04;C07D413/04;C07D417/04;C07D471/04;C07D471/06;C07D471/16;C07D487/04;C07D487/10;C07D498/06;C07D498/16;C07D519/00 主分类号 C07D239/92
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