发明名称 PROCESS FOR MAKING SUBSTITUTED PYRAZOLES
摘要 This invention is directed to a process for making substituted pyrazoles, (I) tautomers of the substituted pyrazoles, and salts of the substituted pyrazoles and tautomers, wherein R3A, R3B, R3C, Y1, Y2, Y3, Y4, and Y5 are as defined in the specification. The process comprises: forming a mixture by a process comprising introducing a hydrazone (II) and an optionally-substituted benzoyl halide (III) into a reactor, and heating the mixture to a temparature of greater than 50 °C (II); and (III).
申请公布号 YU30504(A) 申请公布日期 2006.08.17
申请号 YU2004P000305 申请日期 2002.09.25
申请人 PHARMACIA CORPORATION 发明人 ALLEN, KIMBERLEY;ANDERSON, DENNIS;BALDUS, JOHN;CLARK, JERRY;DUKESHERER, DAN;EDNEY, ALBERT;LAU, PATRICK;MAO, MICHAEL;MCDERMOTT, LISA;MOE, JODIE;MUDIPALLI, PARTHA;NAING, WIN;SCHILKE, TOBIN;SELNESS, SHAUN;SEYMOUR, CHRISTINE;VISWANATH, SHEKHAR;WALKER, JOHN;YALAMANCHILI, GOPICHAND
分类号 C07D403/14;A61K31/506;A61P1/04;A61P1/16;A61P3/10;A61P9/00;A61P9/04;A61P9/10;A61P13/12;A61P15/00;A61P17/00;A61P17/02;A61P17/06;A61P19/02;A61P19/10;A61P25/00;A61P25/04;A61P25/14;A61P25/28;A61P27/02;A61P27/06;A61P29/00;A61P31/04;A61P31/16;A61P31/18;A61P31/22;A61P33/06;A61P35/00;A61P37/06;C07D401/14 主分类号 C07D403/14
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