发明名称 |
PROCESS FOR MAKING SUBSTITUTED PYRAZOLES |
摘要 |
This invention is directed to a process for making substituted pyrazoles, (I) tautomers of the substituted pyrazoles, and salts of the substituted pyrazoles and tautomers, wherein R3A, R3B, R3C, Y1, Y2, Y3, Y4, and Y5 are as defined in the specification. The process comprises: forming a mixture by a process comprising introducing a hydrazone (II) and an optionally-substituted benzoyl halide (III) into a reactor, and heating the mixture to a temparature of greater than 50 °C (II); and (III). |
申请公布号 |
YU30504(A) |
申请公布日期 |
2006.08.17 |
申请号 |
YU2004P000305 |
申请日期 |
2002.09.25 |
申请人 |
PHARMACIA CORPORATION |
发明人 |
ALLEN, KIMBERLEY;ANDERSON, DENNIS;BALDUS, JOHN;CLARK, JERRY;DUKESHERER, DAN;EDNEY, ALBERT;LAU, PATRICK;MAO, MICHAEL;MCDERMOTT, LISA;MOE, JODIE;MUDIPALLI, PARTHA;NAING, WIN;SCHILKE, TOBIN;SELNESS, SHAUN;SEYMOUR, CHRISTINE;VISWANATH, SHEKHAR;WALKER, JOHN;YALAMANCHILI, GOPICHAND |
分类号 |
C07D403/14;A61K31/506;A61P1/04;A61P1/16;A61P3/10;A61P9/00;A61P9/04;A61P9/10;A61P13/12;A61P15/00;A61P17/00;A61P17/02;A61P17/06;A61P19/02;A61P19/10;A61P25/00;A61P25/04;A61P25/14;A61P25/28;A61P27/02;A61P27/06;A61P29/00;A61P31/04;A61P31/16;A61P31/18;A61P31/22;A61P33/06;A61P35/00;A61P37/06;C07D401/14 |
主分类号 |
C07D403/14 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|