发明名称 AZACYCLIC COMPOUNDS AS INHIBITORS OF SENSORY NEURONE SPECIFIC CHANNELS ( SNS )
摘要 Compounds of the formula (I) , and pharmaceutically acceptable salts thereof , are found to be antagonists of SNS sodium channels. They are therefore useful as analgesic and neuroprotective agents. wherein: - Ar represents a phenyl ring or a 5 - to 6- membered heteroaryl group; - m is 1 , 2 or 3 .
申请公布号 WO2006082354(A1) 申请公布日期 2006.08.10
申请号 WO2006GB00040 申请日期 2006.01.06
申请人 VERNALIS (R & D) LIMITED;HAMLYN, RICHARD;HUCKSTEP, MIKE;EARNSHAW, CHRISTOPHER, GEOFFREY;STOKES, STEPHEN;TICKLE, DAVID;ALLART, BRIGITTE;BOYD, JOSEPH, WILLIAM;KNUTSEN, LARS, JACOB, STRAY;LYNCH, ROSEMARY;PATIENT, LEE 发明人 HAMLYN, RICHARD;HUCKSTEP, MIKE;EARNSHAW, CHRISTOPHER, GEOFFREY;STOKES, STEPHEN;TICKLE, DAVID;ALLART, BRIGITTE;BOYD, JOSEPH, WILLIAM;KNUTSEN, LARS, JACOB, STRAY;LYNCH, ROSEMARY;PATIENT, LEE
分类号 C07D217/04;A61K31/4035;A61K31/4365;A61K31/472;A61K31/4725;A61K31/538;A61K31/5415;A61P25/04;A61P25/06;C07D209/48;C07D401/12;C07D405/12;C07D413/04;C07D413/06;C07D417/04;C07D417/06;C07D495/04 主分类号 C07D217/04
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