发明名称 NOVEL MCH RECEPTOR ANTAGONISTS
摘要 The present invention relates to a melanin concentrating hormone antagonist compound of formula (I); wherein Ar<SUP>1</SUP>, L<SUB>1</SUB>, R<SUP>1</SUP>, q, X, R<SUP>2</SUP>, R<SUP>3</SUP>, R<SUP>4</SUP>, and R<SUP>5</SUP> are as defined, or a pharmaceutically acceptable salt, solvate, or enantiomer thereof useful in the treatment, prevention or amelioration of symptoms associated with obesity and related diseases.
申请公布号 WO2006066173(A3) 申请公布日期 2006.07.27
申请号 WO2005US45864 申请日期 2005.12.16
申请人 ELI LILLY AND COMPANY;BECK, JAMES, PETER;WAKEFIELD, BRIAN, DAVID;CORDIER, FREDERIC, LAURENT;DOMINGUEZ-MANZANARES, ESTEBAN;GARDINIER, KEVIN, MATTHEW;GREENEN, PETER, MICHAEL;SAVIN, KENNETH, ALLEN 发明人 BECK, JAMES, PETER;WAKEFIELD, BRIAN, DAVID;CORDIER, FREDERIC, LAURENT;DOMINGUEZ-MANZANARES, ESTEBAN;GARDINIER, KEVIN, MATTHEW;GREENEN, PETER, MICHAEL;SAVIN, KENNETH, ALLEN
分类号 C07D417/04;A61K31/41;A61K31/435;A61K31/495;A61P3/04;A61P3/06;A61P3/10;C07D263/58;C07D277/68;C07D277/82;C07D413/04;C07D413/12;C07D417/14 主分类号 C07D417/04
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