发明名称 SALT FORMS OF 4-(4-METHYLPIPERAZIN-1-YLMETHYL)-n-[4-METHYL-3-(4-PYRIDIN-3-YL)PYRIMIDIN-2-YLAMINO)PHENYL]-BENZAMIDE
摘要 The present invention relates to acid addition salts of 4-[4-methyl-1-piperazinylmethyl]-N-[4-methyl-3-[[4-¢3-pyridinyl-2-pyrimidinyl]amino]phenyl]-benzamide, which are selected from the group consisting of a tartrate salt, such as a (D)(-) tartrate salt or a (L)(+) tartrate salt, a hydrochloride salt, a citrate sat, a malate salt, a fumarate salt, a succinate salt, a benzoate salt, a benzenesulfonate salt, a pamoate salt, a formate salt, a malonate salt, a 1,5-naphthalenedisulfonate salt, a salicylate salt, a cyclohexanesulfamate salt, a lactate salt, a mandelate salt, aq glutarate salt, an adipate salt, a squarate salt, a vanillate salt, an oxaloacetate salt, an ascorbate salt and a sulfate salt.
申请公布号 WO2005075454(A3) 申请公布日期 2006.07.27
申请号 WO2005EP01077 申请日期 2005.02.03
申请人 NOVARTIS AG;NOVARTIS PHARMA GMBH;BUERGER, HANS, MICHAEL;MANLEY, PAUL, WILLIAM;MUTZ, MICHAEL 发明人 BUERGER, HANS, MICHAEL;MANLEY, PAUL, WILLIAM;MUTZ, MICHAEL
分类号 C07D401/04;A61K31/505;A61P35/02 主分类号 C07D401/04
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