发明名称 DIPEPTIDYL PEPTIDASE INHIBITORS
摘要 Compounds, pharmaceutical compositions, kits and methods ar provided for use with DPP-IV and other S9 proteases that comprise a compond of the formula: (I) wherein R<SUB>2 </SUB>is amino (C<SUB>1-6</SUB>)alkyl, hetero(C<SUB>3-12</SUB>)cycloalkyl, hetero(C<SUB>4-12</SUB>)bicycloaryl, heteroaryl, or cyano; and W, X, Y, Z, R<SUB>1</SUB>, R<SUB>5</SUB> and R<SUB>7</SUB> are as defined herein.
申请公布号 WO2006020017(A3) 申请公布日期 2006.07.27
申请号 WO2005US25153 申请日期 2005.07.15
申请人 TAKEDA PHARMACEUTICAL COMPANY LIMITED;FENG, JUN;GWALTNEY, STEVEN;LAM, BETTY;ZHANG, ZHIYUAN 发明人 FENG, JUN;GWALTNEY, STEVEN;LAM, BETTY;ZHANG, ZHIYUAN
分类号 C07D471/04;A61K31/519;C07D471/14 主分类号 C07D471/04
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