发明名称 |
DIPEPTIDYL PEPTIDASE INHIBITORS |
摘要 |
Compounds, pharmaceutical compositions, kits and methods ar provided for use with DPP-IV and other S9 proteases that comprise a compond of the formula: (I) wherein R<SUB>2 </SUB>is amino (C<SUB>1-6</SUB>)alkyl, hetero(C<SUB>3-12</SUB>)cycloalkyl, hetero(C<SUB>4-12</SUB>)bicycloaryl, heteroaryl, or cyano; and W, X, Y, Z, R<SUB>1</SUB>, R<SUB>5</SUB> and R<SUB>7</SUB> are as defined herein. |
申请公布号 |
WO2006020017(A3) |
申请公布日期 |
2006.07.27 |
申请号 |
WO2005US25153 |
申请日期 |
2005.07.15 |
申请人 |
TAKEDA PHARMACEUTICAL COMPANY LIMITED;FENG, JUN;GWALTNEY, STEVEN;LAM, BETTY;ZHANG, ZHIYUAN |
发明人 |
FENG, JUN;GWALTNEY, STEVEN;LAM, BETTY;ZHANG, ZHIYUAN |
分类号 |
C07D471/04;A61K31/519;C07D471/14 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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