发明名称 |
N-BIARYLMETHYL AMINOCYCLOALKANECARBOXAMIDE DERIVATIVES |
摘要 |
N-Biarylmethylaminocycloalkanecarboxamide derivatives are bradykinin B1 antagonists or inverse agonists useful in the treatment or prevention of symptoms such as pain and inflammation associated with the bradykinin B1 pathway. |
申请公布号 |
ZA200500471(B) |
申请公布日期 |
2006.07.26 |
申请号 |
ZA20050000471 |
申请日期 |
2005.01.18 |
申请人 |
MERCK & CO INC., A CORPORATION ORGANIZED UNDER THE LAWS OF THE STATE OF NEW JERSEY, UNITED STATES OF AMERICA |
发明人 |
Michael R WOOD;Scott D KUDUK;MARK G BOCK |
分类号 |
A61K;C07D213/24;A61K31/44;A61K31/4439;A61K31/505;A61K31/506;A61P1/04;A61P1/16;A61P1/18;A61P3/10;A61P7/10;A61P9/00;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P13/10;A61P13/12;A61P17/00;A61P17/02;A61P17/06;A61P19/02;A61P19/06;A61P21/00;A61P25/00;A61P25/04;A61P25/06;A61P25/28;A61P27/02;A61P29/00;A61P31/04;A61P37/08;C07D;C07D213/40;C07D213/56;C07D213/61;C07D239/02;C07D239/28;C07D239/42;C07D401/10;C07D401/12;C07D401/14;C07D413/10;C07D413/12;C07D417/12 |
主分类号 |
A61K |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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