发明名称 N-BIARYLMETHYL AMINOCYCLOALKANECARBOXAMIDE DERIVATIVES
摘要 N-Biarylmethylaminocycloalkanecarboxamide derivatives are bradykinin B1 antagonists or inverse agonists useful in the treatment or prevention of symptoms such as pain and inflammation associated with the bradykinin B1 pathway.
申请公布号 ZA200500471(B) 申请公布日期 2006.07.26
申请号 ZA20050000471 申请日期 2005.01.18
申请人 MERCK & CO INC., A CORPORATION ORGANIZED UNDER THE LAWS OF THE STATE OF NEW JERSEY, UNITED STATES OF AMERICA 发明人 Michael R WOOD;Scott D KUDUK;MARK G BOCK
分类号 A61K;C07D213/24;A61K31/44;A61K31/4439;A61K31/505;A61K31/506;A61P1/04;A61P1/16;A61P1/18;A61P3/10;A61P7/10;A61P9/00;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P13/10;A61P13/12;A61P17/00;A61P17/02;A61P17/06;A61P19/02;A61P19/06;A61P21/00;A61P25/00;A61P25/04;A61P25/06;A61P25/28;A61P27/02;A61P29/00;A61P31/04;A61P37/08;C07D;C07D213/40;C07D213/56;C07D213/61;C07D239/02;C07D239/28;C07D239/42;C07D401/10;C07D401/12;C07D401/14;C07D413/10;C07D413/12;C07D417/12 主分类号 A61K
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