发明名称 |
METHOD FOR PREPARATION OF 10,11-DIHYDRO-10-HYDROXY-5H-DIBENZ/B,F/AZEPINE-5-CARBOXAMIDE |
摘要 |
A process for the preparation of 10,11-dihydro-10-hydroxy-5H-dibenz/b,f/azepine-5-carboxamide (1) by ring opening of 11a,10b-dihydro-6H-dibenz/b,f/oxireno[d]azepine-6-carboxamide (5), characterised in that the ring opening is carried out under conditions of elevated pressure. |
申请公布号 |
WO2006075925(A2) |
申请公布日期 |
2006.07.20 |
申请号 |
WO2006PT00002 |
申请日期 |
2006.01.13 |
申请人 |
PORTELA & C.A., S.A.;LEARMONTH, DAVID, ALEXANDER;WEINGAERTNER, GUENTER;KRAEMER, MATTHIAS |
发明人 |
LEARMONTH, DAVID, ALEXANDER;WEINGAERTNER, GUENTER;KRAEMER, MATTHIAS |
分类号 |
C07D223/22;A61K31/55;C07D491/04 |
主分类号 |
C07D223/22 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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