发明名称 METHOD FOR PREPARATION OF 10,11-DIHYDRO-10-HYDROXY-5H-DIBENZ/B,F/AZEPINE-5-CARBOXAMIDE
摘要 A process for the preparation of 10,11-dihydro-10-hydroxy-5H-dibenz/b,f/azepine-5-carboxamide (1) by ring opening of 11a,10b-dihydro-6H-dibenz/b,f/oxireno[d]azepine-6-carboxamide (5), characterised in that the ring opening is carried out under conditions of elevated pressure.
申请公布号 WO2006075925(A2) 申请公布日期 2006.07.20
申请号 WO2006PT00002 申请日期 2006.01.13
申请人 PORTELA & C.A., S.A.;LEARMONTH, DAVID, ALEXANDER;WEINGAERTNER, GUENTER;KRAEMER, MATTHIAS 发明人 LEARMONTH, DAVID, ALEXANDER;WEINGAERTNER, GUENTER;KRAEMER, MATTHIAS
分类号 C07D223/22;A61K31/55;C07D491/04 主分类号 C07D223/22
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