发明名称 5-MEMBERED ANNELATED HETEROCYCLIC PYRIMIDINES AS KINASE INHIBITORS
摘要 This invention comprises the novel compounds of formula (I) wherein R1, R2, R3, R4, R5, R6, Q1, Q2, X1, X2, Y and Z have defined meanings, having cell cycle kinase inhibiting enzymatic activity, their preparation, compositions containing them and their use as a medicine.
申请公布号 CA2594425(A1) 申请公布日期 2006.07.20
申请号 CA20062594425 申请日期 2006.01.09
申请人 JANSSEN PHARMACEUTICA NAAMLOZE VENNOOTSCHAP 发明人 LARDEAU, DELPHINE YVONNE RAYMONDE;LIGNY, YANNICK AIME EDDY;TEN HOLTE, PETER;PERERA, TIMOTHY PIETRO SUREN;LAVRIJSSEN, TOM;FREYNE, EDDY JEAN EDGARD;LACRAMPE, JEAN FERNAND ARMAND
分类号 C07D473/32;A61K31/519;A61K31/52;A61P35/00;C07D487/04 主分类号 C07D473/32
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