发明名称 |
5-MEMBERED ANNELATED HETEROCYCLIC PYRIMIDINES AS KINASE INHIBITORS |
摘要 |
This invention comprises the novel compounds of formula (I) wherein R1, R2, R3, R4, R5, R6, Q1, Q2, X1, X2, Y and Z have defined meanings, having cell cycle kinase inhibiting enzymatic activity, their preparation, compositions containing them and their use as a medicine.
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申请公布号 |
CA2594425(A1) |
申请公布日期 |
2006.07.20 |
申请号 |
CA20062594425 |
申请日期 |
2006.01.09 |
申请人 |
JANSSEN PHARMACEUTICA NAAMLOZE VENNOOTSCHAP |
发明人 |
LARDEAU, DELPHINE YVONNE RAYMONDE;LIGNY, YANNICK AIME EDDY;TEN HOLTE, PETER;PERERA, TIMOTHY PIETRO SUREN;LAVRIJSSEN, TOM;FREYNE, EDDY JEAN EDGARD;LACRAMPE, JEAN FERNAND ARMAND |
分类号 |
C07D473/32;A61K31/519;A61K31/52;A61P35/00;C07D487/04 |
主分类号 |
C07D473/32 |
代理机构 |
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代理人 |
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地址 |
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