发明名称 QUINOLINES AND QUINAZOLINE ANALOGS AND THEIR USE AS MEDICAMENTS FOR TREATING CANCER
摘要 Selected compounds of Formula (I) are effective for prophylaxis and treatment of diseases, such as HGF mediated diseases such as cancer and the like. The subject invention also relates to processes for making such compounds as well as to intermediates useful in such processes. R - X - W - A - Y - R Formula (I) wherein R is X is O, S, NR2 or CR3R4 W is an substituted or unsubstituted aryl or substituted or unsubstituted 5- or 6- membered heteroaryl.
申请公布号 WO2006060318(A3) 申请公布日期 2006.07.20
申请号 WO2005US42935 申请日期 2005.11.29
申请人 AMGEN INC.;KIM, TAE-SEONG;BELLON, STEVEN;BOOKER, SHON;D'ANGELO, NOEL;DOMINGUEZ, CELIA;FELLOWS, INGRID;LEE, MATTHEW;LIU, LONGBIN;RAINBEAU, ELIZABETH;SIEGMUND, AARON, C.;TASKER, ANDREW;XI, NING;CHENG, YUAN 发明人 KIM, TAE-SEONG;BELLON, STEVEN;BOOKER, SHON;D'ANGELO, NOEL;DOMINGUEZ, CELIA;FELLOWS, INGRID;LEE, MATTHEW;LIU, LONGBIN;RAINBEAU, ELIZABETH;SIEGMUND, AARON, C.;TASKER, ANDREW;XI, NING;CHENG, YUAN
分类号 A61K31/4709;A61P35/00;C07D401/12;C07D401/14 主分类号 A61K31/4709
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