发明名称 5-MEMBERED ANNELATED HETEROCYCLIC PYRIMIDINES AS KINASE INHIBITORS
摘要 <p>This invention comprises the novel compounds of formula (I) wherein R&lt;SUP&gt;1&lt;/SUP&gt;, R&lt;SUP&gt;2&lt;/SUP&gt;, R&lt;SUP&gt;3&lt;/SUP&gt;, R&lt;SUP&gt;4&lt;/SUP&gt;, R&lt;SUP&gt;5&lt;/SUP&gt;, R&lt;SUP&gt;6&lt;/SUP&gt;, Q&lt;SUP&gt;1&lt;/SUP&gt;, Q&lt;SUP&gt;2&lt;/SUP&gt;, X&lt;SUP&gt;1&lt;/SUP&gt;, X&lt;SUP&gt;2&lt;/SUP&gt;, Y and Z have defined meanings, having cell cycle kinase inhibiting enzymatic activity, their preparation, compositions containing them and their use as a medicine.</p>
申请公布号 WO2006074985(A1) 申请公布日期 2006.07.20
申请号 WO2006EP50097 申请日期 2006.01.09
申请人 JANSSEN PHARMACEUTICA N.V.;FREYNE, EDDY, JEAN, EDGARD;LACRAMPE, JEAN, FERNAND, ARMAND;PERERA, TIMOTHY, PIETRO, SUREN;TEN HOLTE, PETER;LIGNY, YANNICK, AIME, EDDY;LARDEAU, DELPHINE, YVONNE, RAYMONDE;LAVRIJSSEN, TOM 发明人 FREYNE, EDDY, JEAN, EDGARD;LACRAMPE, JEAN, FERNAND, ARMAND;PERERA, TIMOTHY, PIETRO, SUREN;TEN HOLTE, PETER;LIGNY, YANNICK, AIME, EDDY;LARDEAU, DELPHINE, YVONNE, RAYMONDE;LAVRIJSSEN, TOM
分类号 C07D473/32;A61K31/519;A61K31/52;A61P35/00;C07D487/04 主分类号 C07D473/32
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