发明名称 5-phenypyrimidines their preparation compositions comprising them and their use
摘要 5-Phenylpyrimidines of the formula I in which the substituents and the index are as defined below: R<SUP>1</SUP>,R<SUP>2 </SUP>are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl, and R<SUP>1 </SUP>and R<SUP>2 </SUP>together with the nitrogen atom to which they are attached may also form a saturated or unsaturated ring which may be interrupted by an ether, thio, sulfoxyl or sulfonyl group and may be substituted by one to four groups R<SUP>a </SUP>and/or R<SUP>b</SUP>; R<SUP>3 </SUP>is hydrogen, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy or alkenyloxy; R<SUP>4 </SUP>is hydrogen, halogen, cyano, hydroxyl, mercapto, azido, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, -ON-CR<SUP>a</SUP>R<SUP>b</SUP>, -CR<SUP>c</SUP>-NOR<SUP>a</SUP>, -NR<SUP>c</SUP>N-CR<SUP>a</SUP>R<SUP>b</SUP>, -NR<SUP>a</SUP>R<SUP>b</SUP>, -NR<SUP>c</SUP>NR<SUP>a</SUP>R<SUP>b</SUP>, -NOR<SUP>a</SUP>, -NR<SUP>c</SUP>C(-NR<SUP>c'</SUP>)NR<SUP>a</SUP>R<SUP>b</SUP>, -NR<SUP>c</SUP>C(-O)NR<SUP>a</SUP>R<SUP>b</SUP>, -NR<SUP>a</SUP>C(-O)R<SUP>c</SUP>, -NR<SUP>a</SUP>C(-NOR<SUP>c</SUP>)R<SUP>c'</SUP>, -OC(-O)R<SUP>c</SUP>, -C(-NOR<SUP>c</SUP>)NR<SUP>a</SUP>R<SUP>b</SUP>, -CR<SUP>c</SUP>(-NNR<SUP>a</SUP>R<SUP>b</SUP>), -C(-O)NR<SUP>a</SUP>R<SUP>b </SUP>or -C(-O)R<SUP>c</SUP>; in which R<SUP>a</SUP>, R<SUP>b </SUP>and R<SUP>c </SUP>are as defined in the description; X is halogen, alkyl, alkoxy or haloalkyl; and m is an integer from 1 to 5; processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.
申请公布号 US2006148764(A1) 申请公布日期 2006.07.06
申请号 US20040495280 申请日期 2004.05.11
申请人 GYPSER ANDREAS 发明人 GYPSER ANDREAS
分类号 A61K31/655;A01N43/54;A61K31/505;A61K31/506;A61K31/513;C07D239/42;C07D239/46;C07D239/47;C07D239/48;C07D239/52;C07D401/06;C07D401/14;C07D403/02;C07D403/12 主分类号 A61K31/655
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