发明名称 PYRIMIDINE DERIVATIVES AS GPCR AGONISTS
摘要 <p>Compounds of formula (I): R&lt;SUP&gt;1&lt;/SUP&gt;-A-V-B-R&lt;SUP&gt;2&lt;/SUP&gt; , wherein V is phenyl or a 6-membered heteroaryl ring containing up to three N-atoms, or pharmaceutically acceptable salts thereof, are agonists of GPR116 and are useful for the treatment of obesity, and for the treatment of diabetes.</p>
申请公布号 WO2006070208(A1) 申请公布日期 2006.07.06
申请号 WO2005GB50266 申请日期 2005.12.30
申请人 PROSIDION LTD.;BRADLEY, STUART, EDWARD;FYFE, MATTHEW, COLIN, THOR;THOMAS, GERARD, HUGH 发明人 BRADLEY, STUART, EDWARD;FYFE, MATTHEW, COLIN, THOR;THOMAS, GERARD, HUGH
分类号 C07D401/14;A61K31/495;A61P3/00 主分类号 C07D401/14
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