发明名称 Process for preparing 5,6-dihydro-4-(S)-(ethylamino)-6-(S) methyl-4H-thieno[2,3b]thiopyran-2-sulphonamide-7,7-dioxide HCI
摘要 The present invention relates to an improved process for the preparation of 5,6-dihydro-4-(S)-(ethylamino)-6-(S)methyl-4H-thieno[2,3b]thiopyran-2-sulphonamide-7,7-dioxide hydrochloride of formula (I) commonly known as Dorzolamide Hydrochloride useful as an agent to reduce intraoccular pressure by inhibiting carbonic anhydrase enzyme
申请公布号 US2006142595(A1) 申请公布日期 2006.06.29
申请号 US20040024029 申请日期 2004.12.28
申请人 COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH 发明人 GURJAR MUKUND K.;DESHMUKH MADHUSUDAN N.;PAUL VINCENT;TARUR VENKATASUBRAMANIAN R.;SATHE DHANANJAY G.;PARDESHI SANTOSH P.;NAIK SANJAY J.;NAIK TUSHAR A.
分类号 C07D495/02 主分类号 C07D495/02
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