发明名称 |
Substituted hydroxyethylamines |
摘要 |
This present invention relates to prodrug compounds of the formula (Y) and pharmaceutical salts thereof: where RN, R1, R2, R3R4 and RC are defined herein, which are useful in treating Alzheimer's disease and other similar diseases. |
申请公布号 |
ZA200406791(B) |
申请公布日期 |
2006.06.28 |
申请号 |
ZA20040006791 |
申请日期 |
2004.08.26 |
申请人 |
ELAN PHARMACEUTICALS, INC.;PHARMACIA & UPJOHN COMPANY |
发明人 |
JOHN VARGEHESE;JAGODZINSKA BARBARA;MAILLARD MICHEL;BECK JAMES P;TENBRINK RUTH E;GETMAN DANIEL |
分类号 |
C07D295/12;A61K;A61K31/132;A61K31/137;A61K31/165;A61K31/166;A61K31/195;A61K31/215;A61K31/325;A61K31/33;A61K31/341;A61K31/36;A61K31/381;A61K31/40;A61K31/4045;A61K31/41;A61K31/415;A61K31/417;A61K31/42;A61K31/421;A61K31/423;A61K31/4245;A61K31/426;A61K31/429;A61K31/433;A61K31/44;A61K31/4402;A61K31/4406;A61K31/4409;A61K31/455;A61K31/495;A61K31/4965;A61K31/50;A61K31/505;A61K31/5375;A61K47/48;A61P;A61P25/16;A61P25/28;C07C;C07C217/58;C07C233/78;C07C247/10;C07C247/12;C07C255/57;C07C271/16;C07C271/20;C07C311/16;C07D;C07D207/09;C07D207/335;C07D207/48;C07D209/14;C07D211/58;C07D213/36;C07D213/71;C07D213/81;C07D213/82;C07D213/89;C07D231/12;C07D231/16;C07D233/64;C07D233/84;C07D237/08;C07D239/26;C07D241/12;C07D257/04;C07D261/10;C07D261/18;C07D263/32;C07D263/46;C07D263/48;C07D263/58;C07D271/06;C07D271/10;C07D277/20;C07D277/28;C07D277/36;C07D285/08;C07D285/12;C07D295/20;C07D295/205;C07D295/22;C07D295/26;C07D307/14;C07D307/20;C07D307/52;C07D307/64;C07D317/58;C07D333/20;C07D333/28;C07D333/34;C07D333/38;C07D333/40;C07D513/04 |
主分类号 |
C07D295/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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